Reaction Details |
| Report a problem with these data |
Target | Caspase-1 |
---|
Ligand | BDBM10246 |
---|
Substrate/Competitor | Caspase-7 Fluorometric Substrate Ac-Asp-Glu-Val-Asp-AFC |
---|
Meas. Tech. | Fluorometric Assay |
---|
pH | 7.5±n/a |
---|
Temperature | 298.15±n/a K |
---|
Ki | 18±n/a nM |
---|
Citation | Garcia-Calvo, M; Peterson, EP; Leiting, B; Ruel, R; Nicholson, DW; Thornberry, NA Inhibition of human caspases by peptide-based and macromolecular inhibitors. J Biol Chem273:32608-13 (1998) [PubMed] Article |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
Caspase-1 |
---|
Name: | Caspase-1 |
Synonyms: | CASP1 | CASP1_HUMAN | Caspase | Caspase 1 | ICE | IL1BC | IL1BCE | Interleukin-1 beta convertase | Interleukin-1 beta-converting enzyme |
Type: | Enzyme |
Mol. Mass.: | 45154.13 |
Organism: | Homo sapiens (Human) |
Description: | P29466 |
Residue: | 404 |
Sequence: | MADKVLKEKRKLFIRSMGEGTINGLLDELLQTRVLNKEEMEKVKRENATVMDKTRALIDS
VIPKGAQACQICITYICEEDSYLAGTLGLSADQTSGNYLNMQDSQGVLSSFPAPQAVQDN
PAMPTSSGSEGNVKLCSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRT
GAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIR
EGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKDSVG
VSGNLSLPTTEEFEDDAIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEY
ACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH
|
|
|
BDBM10246 |
---|
Caspase-7 Fluorometric Substrate Ac-Asp-Glu-Val-Asp-AFC |
---|
Name: | Caspase-7 Fluorometric Substrate Ac-Asp-Glu-Val-Asp-AFC |
Synonyms: | Ac-DEVD-AFC | Ac-DEVD-AMC | Fluorometric Tetrapeptide Ac-DEVD-AMC |
Type: | Peptide |
Mol. Mass.: | 473.41 |
Organism: | n/a |
Description: | Molecular Mass of DEVD |
Residue: | 4 |
Sequence: | |