| Reaction Details |
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 | Report a problem with these data |
| Target | C-C chemokine receptor type 9 |
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| Ligand | BDBM393600 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | FLIPR Assay |
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| Ki | 4.00±n/a nM |
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| Citation |  Bakthavatchalam, R; Basu, MK; Behera, AK; Venkateshappa, C; Hewson, CA; Kadnur, SV; Kalindjian, SB; Kulkarni, B; Saxena, R; Suresh, J; Viswanathan, V; Zainuddin, M; Dharshinis, AP; Kristam, R Compounds useful as CCR9 modulators US Patent US9969687 Publication Date 5/15/2018 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| C-C chemokine receptor type 9 |
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| Name: | C-C chemokine receptor type 9 |
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| Synonyms: | CCR9 | CCR9_HUMAN | GPR28 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42023.90 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1510356 |
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| Residue: | 369 |
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| Sequence: | MTPTDFTSPIPNMADDYGSESTSSMEDYVNFNFTDFYCEKNNVRQFASHFLPPLYWLVFI
VGALGNSLVILVYWYCTRVKTMTDMFLLNLAIADLLFLVTLPFWAIAAADQWKFQTFMCK
VVNSMYKMNFYSCVLLIMCISVDRYIAIAQAMRAHTWREKRLLYSKMVCFTIWVLAAALC
IPEILYSQIKEESGIAICTMVYPSDESTKLKSAVLTLKVILGFFLPFVVMACCYTIIIHT
LIQAKKSSKHKALKVTITVLTVFVLSQFPYNCILLVQTIDAYAMFISNCAVSTNIDICFQ
VTQTIAFFHSCLNPVLYVFVGERFRRDLVKTLKNLGCISQAQWVSFTRREGSLKLSSMLL
ETTSGALSL
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|
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| BDBM393600 |
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| n/a |
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| Name | BDBM393600 |
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| Synonyms: | US9969687, Compound 281 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H20ClN3O5S |
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| Mol. Mass. | 485.94 |
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| SMILES | CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(Cl)c2C(=O)N(C(=O)c12)c1ccc[nH]c1=O |
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| Structure | 
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