Reaction Details |
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Target | 3-phosphoinositide-dependent protein kinase 1 [48-359] |
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Ligand | BDBM32450 |
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Substrate/Competitor | Serine/threonine-protein kinase Sgk1 |
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Meas. Tech. | ELISA assay |
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IC50 | 30±n/a nM |
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Citation | Kim, KH; Wissner, A; Floyd, MB; Fraser, HL; Wang, YD; Dushin, RG; Hu, Y; Olland, A; Guo, B; Arndt, K Benzo[c][2,7]naphthyridines as inhibitors of PDK-1. Bioorg Med Chem Lett19:5225-8 (2009) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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3-phosphoinositide-dependent protein kinase 1 [48-359] |
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Name: | 3-phosphoinositide-dependent protein kinase 1 [48-359] |
Synonyms: | 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) | 3-phosphoinositide-dependent protein kinase 1 | PDK1 | PDPK1 | PDPK1_HUMAN | hPDK1 |
Type: | Serine/threonine-protein kinase |
Mol. Mass.: | 35527.50 |
Organism: | Homo sapiens (Human) |
Description: | O15530[48-359] |
Residue: | 312 |
Sequence: | GPAMDGTAAEPRPGAGSLQHAQPPPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSRE
YAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGEL
LKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTA
KVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNE
YLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTW
ENLHQQTPPKLT
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BDBM32450 |
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Serine/threonine-protein kinase Sgk1 |
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Name: | Serine/threonine-protein kinase Sgk1 |
Synonyms: | SGK | SGK1 | SGK1_HUMAN | Serine/threonine-protein kinase Sgk1 | Serine/threonine-protein kinase Sgk1 (SGK) | Serum/glucocorticoid regulated kinase | Serum/glucocorticoid-regulated kinase 1 (SGK1) |
Type: | Other Protein Type |
Mol. Mass.: | 48954.40 |
Organism: | Homo sapiens (Human) |
Description: | Recombinant human SGK-1 enzyme produced in a baculovirus system. |
Residue: | 431 |
Sequence: | MTVKTEAAKGTLTYSRMRGMVAILIAFMKQRRMGLNDFIQKIANNSYACKHPEVQSILKI
SQPQEPELMNANPSPPPSPSQQINLGPSSNPHAKPSDFHFLKVIGKGSFGKVLLARHKAE
EVFYAVKVLQKKAILKKKEEKHIMSERNVLLKNVKHPFLVGLHFSFQTADKLYFVLDYIN
GGELFYHLQRERCFLEPRARFYAAEIASALGYLHSLNIVYRDLKPENILLDSQGHIVLTD
FGLCKENIEHNSTTSTFCGTPEYLAPEVLHKQPYDRTVDWWCLGAVLYEMLYGLPPFYSR
NTAEMYDNILNKPLQLKPNITNSARHLLEGLLQKDRTKRLGAKDDFMEIKSHVFFSLINW
DDLINKKITPPFNPNVSGPNDLRHFDPEFTEEPVPNSIGKSPDSVLVTASVKEAAEAFLG
FSYAPPTDSFL
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