| Reaction Details |
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 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 1 |
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| Ligand | BDBM35414 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing |
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| IC50 | 36972±n/a nM |
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| Citation |  PubChem, PC In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing PubChem Bioassay(2006)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Dual specificity protein phosphatase 1 |
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| Name: | Dual specificity protein phosphatase 1 |
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| Synonyms: | CL100 | DUS1_HUMAN | DUSP1 | Dual specificity protein phosphatase hVH1 | MAP kinase phosphatase 1 | MKP-1 | MKP1 | PTPN10 | Protein-tyrosine phosphatase CL100 | VH1 |
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| Type: | Protein phosphatase |
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| Mol. Mass.: | 39301.48 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4758204 |
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| Residue: | 367 |
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| Sequence: | MVMEVGTLDAGGLRALLGERAAQCLLLDCRSFFAFNAGHIAGSVNVRFSTIVRRRAKGAM
GLEHIVPNAELRGRLLAGAYHAVVLLDERSAALDGAKRDGTLALAAGALCREARAAQVFF
LKGGYEAFSASCPELCSKQSTPMGLSLPLSTSVPDSAESGCSSCSTPLYDQGGPVEILPF
LYLGSAYHASRKDMLDALGITALINVSANCPNHFEGHYQYKSIPVEDNHKADISSWFNEA
IDFIDSIKNAGGRVFVHCQAGISRSATICLAYLMRTNRVKLDEAFEFVKQRRSIISPNFS
FMGQLLQFESQVLAPHCSAEAGSPAMAVLDRGTSTTTVFNFPVSIPVHSTNSALSYLQSP
ITTSPSC
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| BDBM35414 |
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| n/a |
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| Name | BDBM35414 |
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| Synonyms: | 5-oxidanylidene-N3-(oxolan-2-ylmethyl)-N8-pentyl-1-sulfanylidene-4H-[1,3]thiazolo[3,4-a]quinazoline-3,8-dicarboxamide | 5-oxo-3-N-(oxolan-2-ylmethyl)-8-N-pentyl-1-sulfanylidene-4H-[1,3]thiazolo[3,4-a]quinazoline-3,8-dicarboxamide | 5-oxo-N3-(2-oxolanylmethyl)-N8-pentyl-1-sulfanylidene-4H-thiazolo[3,4-a]quinazoline-3,8-dicarboxamide | 5-oxo-N~8~-pentyl-N~3~-(tetrahydrofuran-2-ylmethyl)-1-thioxo-4,5-dihydro[1,3]thiazolo[3,4-a]quinazoline-3,8-dicarboxamide | MLS000094742 | N'-amyl-5-keto-N-(tetrahydrofurfuryl)-1-thioxo-4H-thiazolo[3,4-a]quinazoline-3,8-dicarboxamide | SMR000030295 | cid_3245487 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H26N4O4S2 |
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| Mol. Mass. | 474.596 |
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| SMILES | CCCCCNC(=O)c1ccc2c(c1)n1c([nH]c2=O)c(sc1=S)C(=O)NCC1CCCO1 |
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| Structure | 
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