| Reaction Details |
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 | Report a problem with these data |
| Target | Estrogen receptor |
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| Ligand | BDBM40503 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Estrogen Receptor-alpha Coactivator Binding Potentiators Dose Response Confirmation |
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| EC50 | 23091.6±n/a nM |
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| Citation |  PubChem, PC Estrogen Receptor-alpha Coactivator Binding Potentiators Dose Response Confirmation PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Estrogen receptor |
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| Name: | Estrogen receptor |
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| Synonyms: | ER | ER-alpha | ESR | ESR1 | ESR1_HUMAN | Estradiol receptor | Estrogen receptor | Estrogen receptor (ER alpha) | Estrogen receptor (ER-alpha) | Estrogen receptor alpha (ER alpha) | Estrogen receptor alpha (ER) | NR3A1 | Nuclear receptor subfamily 3 group A member 1 |
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| Type: | Protein |
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| Mol. Mass.: | 66230.44 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P03372 |
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| Residue: | 595 |
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| Sequence: | MTMTLHTKASGMALLHQIQGNELEPLNRPQLKIPLERPLGEVYLDSSKPAVYNYPEGAAY
EFNAAAAANAQVYGQTGLPYGPGSEAAAFGSNGLGGFPPLNSVSPSPLMLLHPPPQLSPF
LQPHGQQVPYYLENEPSGYTVREAGPPAFYRPNSDNRRQGGRERLASTNDKGSMAMESAK
ETRYCAVCNDYASGYHYGVWSCEGCKAFFKRSIQGHNDYMCPATNQCTIDKNRRKSCQAC
RLRKCYEVGMMKGGIRKDRRGGRMLKHKRQRDDGEGRGEVGSAGDMRAANLWPSPLMIKR
SKKNSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINW
AKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEG
MVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLD
KITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLL
LEMLDAHRLHAPTSRGGASVEETDQSHLATAGSTSSHSLQKYYITGEAEGFPATV
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| BDBM40503 |
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| n/a |
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| Name | BDBM40503 |
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| Synonyms: | (3,5-dimethyl-1,2-oxazol-4-yl)methyl 4-methylthieno[2,3-b]indole-2-carboxylate | 4-methyl-2-thieno[2,3-b]indolecarboxylic acid (3,5-dimethyl-4-isoxazolyl)methyl ester | 4-methylthien[2,3-b]indole-2-carboxylic acid (3,5-dimethylisoxazol-4-yl)methyl ester | MLS000098821 | SMR000067420 | cid_2107577 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H16N2O3S |
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| Mol. Mass. | 340.396 |
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| SMILES | Cc1noc(C)c1COC(=O)c1cc2c3ccccc3n(C)c2s1 |
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| Structure | 
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