Ki Summary

Reaction Details

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Target

Sphingosine 1-phosphate receptor 3

Ligand

BDBM31364

Substrate/Competitor

n/a

Meas. Tech.

Dose response cell-based high throughput screening assay for antagonists of the Sphingosine 1-Phosphate Receptor 3 (S1P3)

IC50

3025±n/a nM

Citation

PubChem, PC Dose response cell-based high throughput screening assay for antagonists of the Sphingosine 1-Phosphate Receptor 3 (S1P3) PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Sphingosine 1-phosphate receptor 3

Name:

Sphingosine 1-phosphate receptor 3

Synonyms:

Type:

G Protein-Coupled Receptor (GPCR)

Mol. Mass.:

42278.13

Organism:

Homo sapiens (Human)

Description:

Q99500

Residue:

378

Sequence:

MATALPPRLQPVRGNETLREHYQYVGKLAGRLKEASEGSTLTTVLFLVICSFIVLENLMV
LIAIWKNNKFHNRMYFFIGNLALCDLLAGIAYKVNILMSGKKTFSLSPTVWFLREGSMFV
ALGASTCSLLAIAIERHLTMIKMRPYDANKRHRVFLLIGMCWLIAFTLGALPILGWNCLH
NLPDCSTILPLYSKKYIAFCISIFTAILVTIVILYARIYFLVKSSSRKVANHNNSERSMA
LLRTVVIVVSVFIACWSPLFILFLIDVACRVQACPILFKAQWFIVLAVLNSAMNPVIYTL
ASKEMRRAFFRLVCNCLVRGRGARASPIQPALDPSRSKSSSSNNSSHSPKVKEDLPHTAP
SSCIMDKNAALQNGIFCN

BDBM31364

n/a

Name

BDBM31364

Synonyms:

(1S,2S)-2-Phenyl-cyclopropanecarboxylic acid [1-[5-(4-nitro-phenyl)-furan-2-yl]-meth-(E)-ylidene]-hydrazide | (1S,2S)-N-[[5-(4-nitrophenyl)-2-furanyl]methylideneamino]-2-phenyl-1-cyclopropanecarboxamide | (1S,2S)-N-[[5-(4-nitrophenyl)-2-furyl]methyleneamino]-2-phenyl-cyclopropanecarboxamide | (1S,2S)-N-[[5-(4-nitrophenyl)furan-2-yl]methylideneamino]-2-phenyl-cyclopropane-1-carboxamide | (1S,2S)-N-[[5-(4-nitrophenyl)furan-2-yl]methylideneamino]-2-phenylcyclopropane-1-carboxamide | MLS000332051 | SMR000221450 | cid_16189645

Type

Small organic molecule

Emp. Form.

C21H17N3O4

Mol. Mass.

375.3774

SMILES

[O-][N+](=O)c1ccc(cc1)-c1ccc(\C=N\NC(=O)C2CC2c2ccccc2)o1

Structure