| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein phosphatase |
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| Ligand | BDBM64788 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 5 (PP5) |
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| IC50 | 9572±n/a nM |
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| Citation |  PubChem, PC Fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Serine/threonine-protein phosphatase |
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| Name: | Serine/threonine-protein phosphatase |
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| Synonyms: | H0YDU8_HUMAN | PPP5C | PPP5C protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 55092.68 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_37589898 |
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| Residue: | 484 |
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| Sequence: | MAEGERTECAEPPRDEPPADGALKRAEELKTQANDYFKAKDYENAIKFYSQAIELNPSNA
IYYGNRSLAYLRTECYGYALGDATRAIELDKKYIKGYYRRAASNMALGKFRAALRDYETV
VKVKPHDKDAKMKYQECNKIVKQKAFERAIAGDEHKRSVVDSLDIESMTIEDEYSGPKLE
DGKVTISFMKELMQWYKDQKKLHRKCAYQILVQVKEVLSKLSTLVETTLKETEKITVCGD
THGQFYDLLNIFELNGLPSETNPYIFNGDFVDRGSFSVEVILTLFGFKLLYPDHFHLLRG
NHETDNMNQIYGFEGEVKAKYTAQMYELFSEVFEWLPLAQCINGKVLIMHGGLFSEDGVT
LDDIRKIERNRQPPDSGPMCDLLWSDPQPQNGRSISKRGVSCQFGPDVTKAFLEENNLDY
IIRSHEVKAEGYEVAHGGRCVTVFSAPNYCDQMGNKASYIHLQGSDLRPQFHQFTAVGRP
SSGS
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|
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| BDBM64788 |
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| n/a |
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| Name | BDBM64788 |
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| Synonyms: | 4-[(5-keto-3-methyl-1-phenyl-3-pyrazolin-4-yl)-(4-nitrophenyl)methyl]-5-methyl-2-phenyl-3-pyrazolin-3-one | 5-methyl-4-[(5-methyl-3-oxidanylidene-2-phenyl-1H-pyrazol-4-yl)-(4-nitrophenyl)methyl]-2-phenyl-1H-pyrazol-3-one | 5-methyl-4-[(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-(4-nitrophenyl)methyl]-2-phenyl-1H-pyrazol-3-one | MLS000592130 | SMR000218378 | cid_2251550 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H23N5O4 |
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| Mol. Mass. | 481.5026 |
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| SMILES | Cc1[nH]n(-c2ccccc2)c(=O)c1C(c1c(C)[nH]n(-c2ccccc2)c1=O)c1ccc(cc1)[N+]([O-])=O |
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| Structure | 
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