Reaction Details |
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Target | Pro-thyrotropin-releasing hormone |
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Ligand | BDBM50035057 |
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Substrate/Competitor | n/a |
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Ki | >10000±n/a nM |
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Comments | PDSP_779 |
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Citation | Schipper, J; Tulp, MT; Sijbesma, H Neurochemical profile of eltoprazine. Drug Metabol Drug Interact8:85-114 (1990) [PubMed] Article |
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More Info.: | Get all data from this article |
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Pro-thyrotropin-releasing hormone |
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Name: | Pro-thyrotropin-releasing hormone |
Synonyms: | Prothyroliberin | TRH_RAT | Trh |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 29277.96 |
Organism: | RAT |
Description: | TRH 0 RAT::P01150 |
Residue: | 255 |
Sequence: | MPGPWLLLALALIFTLTGIPESCALPEAAQEEGAVTPDLPGLENVQVRPERRFLWKDLQR
VRGDLGAALDSWITKRQHPGKREEEEKDIEAEERGDLGEGGAWRLHKRQHPGRRANQDKY
SWADEEDSDWMPRSWLPDFFLDSWFSDVPQVKRQHPGRRSFPWMESDVTKRQHPGRRFID
PELQRSWEEKEGEGVLMPEKRQHPGKRALGHPCGPQGTCGQTGLLQLLGDLSRGQETLVK
QSPQVEPWDKEPLEE
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BDBM50035057 |
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n/a |
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Name | BDBM50035057 |
Synonyms: | (eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine | 1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine | CHEMBL282614 | Eltoprazine |
Type | Small organic molecule |
Emp. Form. | C12H16N2O2 |
Mol. Mass. | 220.2676 |
SMILES | C1CN(CCN1)c1cccc2OCCOc12 |
Structure |
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