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TargetPeroxisome proliferator-activated receptor delta
LigandBDBM50304637
Substrate/Competitorn/a
Meas. Tech.ChEBML_1669058
Ki 3.0±n/a nM
Citation Yu, J; Ahn, S; Kim, HJ; Lee, M; Ahn, S; Kim, J; Jin, SH; Lee, E; Kim, G; Cheong, JH; Jacobson, KA; Jeong, LS; Noh, M Polypharmacology of N J Med Chem60:7459-7475 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peroxisome proliferator-activated receptor delta
Name:Peroxisome proliferator-activated receptor delta
Synonyms:NR1C2 | NUC1 | NUCI | Nuclear hormone receptor 1 | Nuclear receptor subfamily 1 group C member 2 | PPAR delta | PPAR-beta | PPARB | PPARD | PPARD_HUMAN | Peroxisome proliferator-activated receptor | Peroxisome proliferator-activated receptor beta | Peroxisome proliferator-activated receptor delta
Type:Enzyme
Mol. Mass.:49910.45
Organism:Homo sapiens (Human)
Description:Q03181
Residue:441
Sequence:
MEQPQEEAPEVREEEEKEEVAEAEGAPELNGGPQHALPSSSYTDLSRSSSPPSLLDQLQM
GCDGASCGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCERSCKIQKK
NRNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTANEGSQYNPQVADLKAFSK
HIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKE
ISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNK
DGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGD
RPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRI
KKTETETSLHPLLQEIYKDMY
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  Blast E-value cutoff:
BDBM50304637
n/a
NameBDBM50304637
Synonyms:9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribofuranosyl)-N6-(3-iodo-benzyl)adenine | CHEMBL596014
TypeSmall organic molecule
Emp. Form.C20H21IN6O3S
Mol. Mass.552.389
SMILESO[C@H]1[C@@H](O)[C@@H](S[C@@H]1C(=O)NC1CC1)n1cnc2c(NCc3cccc(I)c3)ncnc12 |r|
Structure
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