| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet glycoprotein 4 |
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| Ligand | BDBM50242204 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1670776 (CHEMBL4020664) |
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| IC50 | 3600±n/a nM |
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| Citation |  Chignen Possi, K; Mulumba, M; Omri, S; Garcia-Ramos, Y; Tahiri, H; Chemtob, S; Ong, H; Lubell, WD Influences of Histidine-1 and Azaphenylalanine-4 on the Affinity, Anti-inflammatory, and Antiangiogenic Activities of Azapeptide Cluster of Differentiation 36 Receptor Modulators. J Med Chem60:9263-9274 (2017) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet glycoprotein 4 |
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| Name: | Platelet glycoprotein 4 |
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| Synonyms: | Adipocyte membrane protein | CD36_RAT | CD_antigen=CD36 | Cd36 | Fat | Fatty acid translocase | Fatty acid transport protein | GPIIIB | GPIV | Glycoprotein IIIb | PAS IV | PAS-4 | Platelet glycoprotein IV |
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| Type: | PROTEIN |
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| Mol. Mass.: | 52740.95 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_858884 |
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| Residue: | 472 |
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| Sequence: | MGCDRNCGLITGAVIGAVLAVFGGILMPVGDLLIEKTIKREVVLEEGTIAFKNWVKTGTT
VYRQFWIFDVQNPEEVAKNSSKIKVKQRGPYTYRVRYLAKENITQDPKDSTVSFVQPNGA
IFEPSLSVGTENDNFTVLNLAVAAAPHIYTNSFVQGVLNSLIKKSKSSMFQTRSLKELLW
GYKDPFLSLVPYPISTTVGVFYPYNNTVDGVYKVFNGKDNISKVAIIDTYKGKRNLSYWE
SYCDMINGTDAASFPPFVEKSQTLRFFSSDICRSIYAVFESEVNLKGIPVYRFVLPANAF
ASPLQNPDNHCFCTEKVISNNCTSYGVLDIGKCKEGKPVYISLPHFLHASPDVSEPIEGL
NPNEDEHRTYLDVEPITGFTLQFAKRLQVNILVKPARKIEALKNLKRPYIVPILWLNETG
TIGDEKAEMFRNQVTGKIKLLGLVEMVLLGVGVVMFVAFMISYCACRSKNGK
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| BDBM50242204 |
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| n/a |
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| Name | BDBM50242204 |
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| Synonyms: | CHEMBL4086017 |
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| Type | Small organic molecule |
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| Emp. Form. | C43H53BrN12O6 |
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| Mol. Mass. | 913.862 |
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| SMILES | C[C@H](NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)Cc1cnc[nH]1)C(=O)NN(Cc1ccc(Br)cc1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(N)=O |r| |
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| Structure | 
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