| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50002783 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_209762 |
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| Ki | 3.9±n/a nM |
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| Citation |  Ohshima, E; Takami, H; Sato, H; Mohri, S; Obase, H; Miki, I; Ishii, A; Shirakura, S; Karasawa, A; Kubo, K Non-prostanoid thromboxane A2 receptor antagonists with a dibenzoxepin ring system. 2. J Med Chem35:3402-13 (1992) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50002783 |
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| n/a |
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| Name | BDBM50002783 |
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| Synonyms: | 11-[2-(4,6-Dimethyl-benzoimidazol-1-yl)-ethylidene]-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid | CHEMBL324965 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H22N2O3 |
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| Mol. Mass. | 410.4645 |
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| SMILES | Cc1cc(C)c2ncn(C\C=C3/c4ccccc4COc4ccc(cc34)C(O)=O)c2c1 |
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| Structure | 
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