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TargetGag-Pol polyprotein [489-587]
LigandBDBM50421874
Substrate/Competitorn/a
Meas. Tech.ChEBML_159470
IC50 12±n/a nM
Citation Kempf, DJNorbeck, DWCodacovi, LWang, XCKohlbrenner, WEWideburg, NEPaul, DAKnigge, MFVasavanonda, SCraig-Kennard, A Structure-based, C2 symmetric inhibitors of HIV protease. J Med Chem33:2687-9 (1990) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Gag-Pol polyprotein [489-587]
Name:Gag-Pol polyprotein [489-587]
Synonyms:Human immunodeficiency virus type 1 protease | POL_HV1H2 | Pol polyprotein | gag-pol
Type:Enzyme Subunit
Mol. Mass.:10781.16
Organism:Human immunodeficiency virus type 1
Description:P04585[489-587]
Residue:99
Sequence:
PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYD
QILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF
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BDBM50421874
n/a
NameBDBM50421874
Synonyms:CHEMBL2311105
TypeSmall organic molecule
Emp. Form.C31H44N4O5
Mol. Mass.552.7049
SMILESCC(C)[C@H](NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(C)=O)C(C)C
Structure
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