| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50015852 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_209596 |
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| Kd | 8.3±n/a nM |
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| Citation |  Nakane, M; Reid, JA; Han, WC; Das, J; Truc, VC; Haslanger, MF; Garber, D; Harris, DN; Hedberg, A; Ogletree, ML 7-Oxabicyclo[2.2.1]heptyl carboxylic acids as thromboxane A2 antagonists: aza omega-chain analogues. J Med Chem33:2465-76 (1990) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50015852 |
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| n/a |
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| Name | BDBM50015852 |
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| Synonyms: | 7-{3-[(2-Nonanoylamino-acetylamino)-methyl]-7-oxa-bicyclo[2.2.1]hept-2-yl}-hept-5-enoic acid | CHEMBL82146 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H42N2O5 |
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| Mol. Mass. | 450.6114 |
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| SMILES | CCCCCCCCC(=O)NCC(=O)NCC1C2CCC(O2)C1C\C=C\CCCC(O)=O |THB:23:22:21:18.19,15:16:21:18.19| |
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| Structure | 
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