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TargetG-protein coupled receptor 35
LigandBDBM50323327
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1734190 (CHEMBL4149726)
IC50 110±n/a nM
Citation Wei, LHou, TLu, CWang, JZhang, XFang, YZhao, YFeng, JLi, JQu, LPiao, HLLiang, X SAR Studies of  ACS Med Chem Lett9:422-427 (2018) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 35
Name:G-protein coupled receptor 35
Synonyms:G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:34085.57
Organism:Homo sapiens (Human)
Description:gi_33695097
Residue:309
Sequence:
MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
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  Blast E-value cutoff:
BDBM50323327
n/a
NameBDBM50323327
Synonyms:CHEMBL4171772
TypeSmall organic molecule
Emp. Form.C14H8BrCl2N5O
Mol. Mass.413.056
SMILESClc1ccc(C(=O)Nc2cc(Br)ccc2-c2nnn[nH]2)c(Cl)c1
Structure
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