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TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase
LigandBDBM50405938
Substrate/Competitorn/a
Meas. Tech.ChEBML_141590
Ki 800000±n/a nM
Citation Dredar, SABlankenship, JWMarchant, PEManneh, VFries, DS Design and synthesis of inhibitors of N8-acetylspermidine deacetylase. J Med Chem32:984-9 (1989) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
Name:Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
Synonyms:Acetylpolyamine oxidase (APAO) | PAO | PAOX | PAOX_HUMAN | Peroxisomal N(1)-acetyl-spermine/spermidine oxidase | Polyamine oxidase
Type:Enzyme
Mol. Mass.:70274.33
Organism:Homo sapiens (Human)
Description:Q6QHF9
Residue:511
Sequence:
MESTGSVGEAPGGPRVLVVGGGIAGLGAAQRLCGHSAFPHLRVLEATARAGGRIRSERCF
GGVVEVGAHWIHGPSRGNPVFQLAAEYGLLGEKELSQENQLVETGGHVGLPSVSYASSGA
SVSLQLVAEMATLFYGLIDQTREFLHAAETPVPSVGEYLKKEIGQHVAGWTEDEETRKLK
LAVLNSFFNLECCVSGTHSMDLVALAPFGEYTVLPGLDCTFSKGYQGLTNCMMAALPEDT
VVFEKPVKTIHWNGSFQEAAFPGETFPVSVECEDGDRFPAHHVIVTVPLGFLREHLDTFF
DPPLPAEKAEAIRKIGFGTNNKIFLEFEEPFWEPDCQLIQLVWEDTSPLEDAAPELQDAW
FRKLIGFVVLPAFASVHVLCGFIAGLESEFMETLSDEEVLLCLTQVLRRVTGNPRLPAPK
SVLRSRWHSAPYTRGSYSYVAVGSTGGDLDLLAQPLPADGAGAQLQILFAGEATHRTFYS
TTHGALLSGWREADRLLSLWAPQVQQPRPRL
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BDBM50405938
n/a
NameBDBM50405938
Synonyms:CHEMBL81241
TypeSmall organic molecule
Emp. Form.C6H14N2O
Mol. Mass.130.1882
SMILESCC(=O)NCCCCN
Structure
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