Found 20 hits with Last Name = 'fries' and Initial = 'ds' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405943
(CHEMBL176596)Show InChI InChI=1S/C12H26N2O/c1-12(15)8-5-4-6-9-13-10-7-11-14(2)3/h13H,4-11H2,1-3H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405931
(CHEMBL367753)Show InChI InChI=1S/C14H30N2O/c1-4-16(5-2)13-9-12-15-11-8-6-7-10-14(3)17/h15H,4-13H2,1-3H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405937
(CHEMBL173782)Show InChI InChI=1S/C10H22N2O/c1-10(13)6-3-2-4-8-12-9-5-7-11/h12H,2-9,11H2,1H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405942
(CHEMBL175345)Show InChI InChI=1S/C12H24N2O/c1-12(15)6-4-3-5-7-14-10-8-13(2)9-11-14/h3-11H2,1-2H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
| PubMed
| 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405939
(CHEMBL175307)Show InChI InChI=1S/C14H28N2O2/c1-14(17)6-3-2-4-7-15-8-5-9-16-10-12-18-13-11-16/h15H,2-13H2,1H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
| PubMed
| 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50018055
(7-Amino-heptan-2-one | CHEMBL176843)Show InChI InChI=1S/C7H15NO/c1-7(9)5-3-2-4-6-8/h2-6,8H2,1H3 | UniProtKB/SwissProt
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Patents
| PubMed
| 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405932
(CHEMBL176530)Show InChI InChI=1S/C9H20N2O/c1-3-6-10-7-4-5-8-11-9(2)12/h10H,3-8H2,1-2H3,(H,11,12) | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405935
(CHEMBL177305)Show InChI InChI=1S/C8H18N2O/c1-8(11)10-7-5-3-2-4-6-9/h2-7,9H2,1H3,(H,10,11) | UniProtKB/SwissProt
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405928
(CHEMBL174669)Show InChI InChI=1S/C10H22N2O/c1-10(13)12-9-7-5-3-2-4-6-8-11/h2-9,11H2,1H3,(H,12,13) | UniProtKB/SwissProt
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 7.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405940
(CHEMBL177890)Show InChI InChI=1S/C12H26N2O/c1-12(15)14-11-9-7-5-3-2-4-6-8-10-13/h2-11,13H2,1H3,(H,14,15) | UniProtKB/SwissProt
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 1.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405930
(CHEMBL174887)Show InChI InChI=1S/C8H17ClN2O/c9-7-8(12)11-6-4-2-1-3-5-10/h1-7,10H2,(H,11,12) | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
| PubMed
| 1.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405934
(CHEMBL176764)Show InChI InChI=1S/C10H22N2O2/c1-14-10(13)12-9-7-5-3-2-4-6-8-11/h2-9,11H2,1H3,(H,12,13) | UniProtKB/SwissProt
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 2.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405929
(CHEMBL436093)Show InChI InChI=1S/C7H18N2O2S/c1-12(10,11)9-7-5-3-2-4-6-8/h9H,2-8H2,1H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 3.76E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405941
(CHEMBL177777)Show InChI InChI=1S/C9H22N2O2S/c1-14(12,13)11-9-7-5-3-2-4-6-8-10/h11H,2-10H2,1H3 | UniProtKB/SwissProt
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| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 6.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405938
(CHEMBL81241)Show InChI InChI=1S/C6H14N2O/c1-6(9)8-5-3-2-4-7/h2-5,7H2,1H3,(H,8,9) | UniProtKB/SwissProt
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CHEMBL MCE KEGG PC cid PC sid PDB UniChem
Similars
| PubMed
| 8.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405933
(CHEMBL176800)Show InChI InChI=1S/C9H21N3O/c1-9(13)12-8-4-7-11-6-3-2-5-10/h11H,2-8,10H2,1H3,(H,12,13) | UniProtKB/SwissProt
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CHEMBL MCE KEGG PC cid PC sid PDB UniChem
| PubMed
| 1.37E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase
(Homo sapiens (Human)) | BDBM50405936
(CHEMBL177217)Show InChI InChI=1S/C8H18N2O/c1-2-5-8(11)10-7-4-3-6-9/h2-7,9H2,1H3,(H,10,11) | UniProtKB/SwissProt
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CHEMBL MCE PC cid PC sid UniChem
Similars
| PubMed
| 2.90E+7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific
Curated by ChEMBL
| Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. |
J Med Chem 32: 984-9 (1989)
BindingDB Entry DOI: 10.7270/Q23777PG |
More data for this Ligand-Target Pair | |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223658
(CHEMBL279613)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3/t13-,16+/m0/s1 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223656
(CHEMBL2079647)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223657
(CHEMBL273784)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3/t13?,16-/m0/s1 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
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CHEMBL PC cid PC sid UniChem
Patents
| PubMed
| n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |