| Reaction Details |
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 | Report a problem with these data |
| Target | Melatonin receptor type 1C |
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| Ligand | BDBM50470871 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_104760 (CHEMBL710992) |
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| Ki | 32±n/a nM |
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| Citation |  Mathé-Allainmat, M; Gaudy, F; Sicsic, S; Dangy-Caye, AL; Shen, S; Brémont, B; Benatalah, Z; Langlois, M; Renard, P; Delagrange, P Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors. J Med Chem39:3089-95 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Melatonin receptor type 1C |
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| Name: | Melatonin receptor type 1C |
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| Synonyms: | CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C |
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| Type: | PROTEIN |
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| Mol. Mass.: | 38595.98 |
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| Organism: | Gallus gallus |
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| Description: | ChEMBL_104739 |
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| Residue: | 346 |
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| Sequence: | MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGN
IFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAI
NRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTV
STSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVV
FVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFR
KEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
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| BDBM50470871 |
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| n/a |
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| Name | BDBM50470871 |
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| Synonyms: | CHEMBL106276 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H17NO3 |
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| Mol. Mass. | 271.3111 |
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| SMILES | COc1ccc2ccc(O)c3CC(Cc1c23)NC(C)=O |
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| Structure | 
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