Reaction Details |
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Target | Somatostatin receptor type 5 |
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Ligand | BDBM50474229 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_200989 (CHEMBL857866) |
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Ki | 0.251189±n/a nM |
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Citation | Lewis, I; Bauer, W; Albert, R; Chandramouli, N; Pless, J; Weckbecker, G; Bruns, C A novel somatostatin mimic with broad somatotropin release inhibitory factor receptor binding and superior therapeutic potential. J Med Chem46:2334-44 (2003) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Somatostatin receptor type 5 |
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Name: | Somatostatin receptor type 5 |
Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
Type: | Enzyme |
Mol. Mass.: | 39218.02 |
Organism: | Homo sapiens (Human) |
Description: | P35346 |
Residue: | 364 |
Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
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BDBM50474229 |
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n/a |
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Name | BDBM50474229 |
Synonyms: | CHEMBL3349605 |
Type | Small organic molecule |
Emp. Form. | C59H68N10O10 |
Mol. Mass. | 1077.2322 |
SMILES | [H][C@@]12C[C@H](CN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccc(OCc3ccccc3)cc1)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c3ccccc13)NC(=O)[C@H](Cc1ccc(O)cc1)NC2=O)OC(=O)NCCN |
Structure |
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