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TargetSolute carrier family 22 member 1
LigandBDBM50485613
Substrate/Competitorn/a
Meas. Tech.ChEMBL_836293 (CHEMBL2076306)
IC50 3000±n/a nM
Citation Zhang, LGorset, WDresser, MJGiacomini, KM The interaction of n-tetraalkylammonium compounds with a human organic cation transporter, hOCT1. J Pharmacol Exp Ther288:1192-8 (1999) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Solute carrier family 22 member 1
Name:Solute carrier family 22 member 1
Synonyms:Adrenergic Alpha | OCT1 | Organic cation transporter 1 | S22A1_HUMAN | SLC22A1 | Solute carrier family 22 member 1 | hOCT1
Type:Enzyme Catalytic Domain
Mol. Mass.:61154.85
Organism:Homo sapiens (Human)
Description:Adrenergic Alpha 0 HUMAN::O15245
Residue:554
Sequence:
MPTVDDILEQVGESGWFQKQAFLILCLLSAAFAPICVGIVFLGFTPDHHCQSPGVAELSQ
RCGWSPAEELNYTVPGLGPAGEAFLGQCRRYEVDWNQSALSCVDPLASLATNRSHLPLGP
CQDGWVYDTPGSSIVTEFNLVCADSWKLDLFQSCLNAGFLFGSLGVGYFADRFGRKLCLL
GTVLVNAVSGVLMAFSPNYMSMLLFRLLQGLVSKGNWMAGYTLITEFVGSGSRRTVAIMY
QMAFTVGLVALTGLAYALPHWRWLQLAVSLPTFLFLLYYWCVPESPRWLLSQKRNTEAIK
IMDHIAQKNGKLPPADLKMLSLEEDVTEKLSPSFADLFRTPRLRKRTFILMYLWFTDSVL
YQGLILHMGATSGNLYLDFLYSALVEIPGAFIALITIDRVGRIYPMAMSNLLAGAACLVM
IFISPDLHWLNIIIMCVGRMGITIAIQMICLVNAELYPTFVRNLGVMVCSSLCDIGGIIT
PFIVFRLREVWQALPLILFAVLGLLAAGVTLLLPETKGVALPETMKDAENLGRKAKPKEN
TIYLKVQTSEPSGT
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  Blast E-value cutoff:
BDBM50485613
n/a
NameBDBM50485613
Synonyms:Tetrahexylammonium
TypeSmall organic molecule
Emp. Form.C24H52N
Mol. Mass.354.6758
SMILESCCCCCC[N+](CCCCCC)(CCCCCC)CCCCCC
Structure
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