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Target5-hydroxytryptamine receptor 1B
LigandBDBM50049081
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2025
Ki 2±n/a nM
Citation Glennon RAHong SSBondarev MLaw HDukat MRakhi SPower PFan EKinneau DKamboj RTeitler MHerrick-Davis KSmith C Binding of O-alkyl derivatives of serotonin at human 5-HT1D beta receptors. J Med Chem 39:314-22 (1996) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
5-hydroxytryptamine receptor 1B
Name:Serotonin (5-HT) receptor
Synonyms:5-HT-1B | 5-HT-1D-beta | 5-HT1B | 5-hydroxytryptamine receptor 1B (5-HT1B) | S12 | Serotonin 1D beta receptor | Serotonin Receptor 1B
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:43579.17
Organism:Homo sapiens (Human)
Description:Receptor binding assays were performed using human clone stably expressed in CHO cells
Residue:390
Sequence:
MEEPGAQCAPPPPAGSETWVPQANLSSAPSQNCSAKDYIYQDSISLPWKVLLVMLLALIT
LATTLSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQV
VCDFWLSSDITCCTASILHLCVIALDRYWAITDAVEYSAKRTPKRAAVMIALVWVFSISI
SLPPFFWRQAKAEEEVSECVVNTDHILYTVYSTVGAFYFPTLLLIALYGRIYVEARSRIL
KQTPNRTGKRLTRAQLITDSPGSTSSVTSINSRVPDVPSESGSPVYVNQVKVRVSDALLE
KKKLMAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHLAIFDFFTWLGYL
NSLINPIIYTMSNEDFKQAFHKLIRFKCTS
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  Blast E-value cutoff:
BDBM50049081
n/a
NameBDBM50049081
Synonyms:2-[5-(8,8-Dimethyl-nonyloxy)-1H-indol-3-yl]-ethylamine | CHEMBL107617
TypeSmall organic molecule
Emp. Form.C21H34N2O
Mol. Mass.330.5075
SMILESCC(C)(C)CCCCCCCOc1ccc2[nH]cc(CCN)c2c1
Structure
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