| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50054469 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_46807 (CHEMBL659694) |
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| Ki | 1380±n/a nM |
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| Citation |  Khanolkar, AD; Abadji, V; Lin, S; Hill, WA; Taha, G; Abouzid, K; Meng, Z; Fan, P; Makriyannis, A Head group analogs of arachidonylethanolamide, the endogenous cannabinoid ligand. J Med Chem39:4515-9 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52856.55 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | P20272 |
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| Residue: | 473 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAI
AVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHV
FHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCL
MWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILW
KAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPL
LAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTA
QPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50054469 |
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| n/a |
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| Name | BDBM50054469 |
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| Synonyms: | (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenethioic acid (2-hydroxy-ethyl)-amide | CHEMBL342659 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H37NOS |
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| Mol. Mass. | 363.6 |
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| SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=S)NCCO |
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| Structure | 
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