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TargetCarboxypeptidase G2
LigandBDBM50074672
Substrate/Competitorn/a
Meas. Tech.ChEMBL_45646
Ki 300±n/a nM
Citation Khan THEno-Amooquaye EASearle FBrowne PJOsborn HMBurke PJ Novel inhibitors of carboxypeptidase G2 (CPG2): potential use in antibody-directed enzyme prodrug therapy. J Med Chem 42:951-6 (1999) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Carboxypeptidase G2
Name:Carboxypeptidase G2
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:44005.37
Organism:Pseudomonas aeruginosa
Description:ChEMBL_302801
Residue:412
Sequence:
MHARRLPRLLPLALAFLLSPAAFAADTPAAELLRQAEAERPAYLDTLRQLVAVDSGTGQA
EGLGQLSALLAERLQALGAQVRSAPATPSAGDNLVATLDGTGSKRFLLMIHYDTVFAAGS
AAKRPFREDAERAYGPGVADAKGGVAMVLHALALLRQQGFRDYGRITVLFNPDEETGSAG
SKQLIAELARQQDYVFSYEPPDRDAVTVATNGIDGLLLEVKGRSSHAGSAPEQGRNAILE
LSHQLLRLKDLGDPAKGTTLNWTLARGGEKRNIIPAEASAEADMRYSDPAESERVLADAR
KLTGERLVADTEVSLRLDKGRPPLVKNPASQRLAETAQTLYGRIGKRIEPIAMRFGTDAG
YAYVPGSDKPAVLETLGVVGAGLHSEAEYLELSSIAPRLYLTVALIRELSAD
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  Blast E-value cutoff:
BDBM50074672
n/a
NameBDBM50074672
Synonyms:(R)-2-(4-Methoxy-phenylsulfanylcarbonylamino)-pentanedioic acid | CHEMBL176541
TypeSmall organic molecule
Emp. Form.C13H15NO6S
Mol. Mass.313.326
SMILESCOc1ccc(SC(=O)N[C@H](CCC(O)=O)C(O)=O)cc1
Structure
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