| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50075083 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_225590 |
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| IC50 | 1400±n/a nM |
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| Citation |  Shinozaki, K; Sato, H; Iwakuma, T; Sato, R; Kurimoto, T; Yoshida, K Synthesis and thromboxane A2 antagonistic activity activity of indane derivatives. Bioorg Med Chem Lett9:401-6 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | TA2R_RAT | TXA2/PGH2 | Tbxa2r | Thromboxane A2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36943.05 |
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| Organism: | RAT |
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| Description: | Thromboxane A2 TBXA2R RAT::P34978 |
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| Residue: | 341 |
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| Sequence: | MWLNSTSLGACFRPVNITLQERRAIASPWFAASFCALGLGSNLLALSVLAGARPGAGPRS
SFLALLCGLVLTDFLGLLVTGAVVASQHAALLDWRATDPGCRLCHFMGAAMVFFGLCPLL
LGAAMAAERFVGITRPFSRPAATSRRAWATVGLVWVGAGTLGLLPLLGLGRYSVQYPGSW
CFLTLGAERGDVAFGLMFALLGSVSVGLSLLLNTVSVATLCRVYHAREATQRPRDCEVEM
MVQLVGIMVVATVCWMPLLVFILQTLLQTLPVMSPSGQLLRTTERQLLIYLRVATWNQIL
DPWVYILFRRSVLRRLHPRFTSQLQAVSLHSPPTQAMLSGP
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| BDBM50075083 |
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| n/a |
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| Name | BDBM50075083 |
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| Synonyms: | CHEMBL340073 | Sodium; {2-[(pentane-1-sulfonylamino)-methyl]-indan-5-yl}-acetate |
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| Type | Small organic molecule |
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| Emp. Form. | C17H24NO4S |
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| Mol. Mass. | 338.442 |
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| SMILES | CCCCCS(=O)(=O)NCC1Cc2ccc(CC([O-])=O)cc2C1 |
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| Structure | 
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