| Reaction Details |
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 | Report a problem with these data |
| Target | Cathepsin G |
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| Ligand | BDBM50085366 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_45352 |
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| IC50 | 9300.0±n/a nM |
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| Citation |  Hayashi, Y; Iijima, K; Katada, J; Kiso, Y Structure-activity relationship studies of chloromethyl ketone derivatives for selective human chymase inhibitors. Bioorg Med Chem Lett10:199-201 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Cathepsin G |
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| Name: | Cathepsin G |
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| Synonyms: | CATG_HUMAN | CG | CTSG |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28860.08 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1469016 |
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| Residue: | 255 |
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| Sequence: | MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVL
TAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRR
NRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYD
PRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRT
TMRSFKLLDQMETPL
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| BDBM50085366 |
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| n/a |
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| Name | BDBM50085366 |
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| Synonyms: | CHEMBL292834 | N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(4-methoxy-phenyl)-propionamide |
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| Type | Small organic molecule |
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| Emp. Form. | C20H22ClNO3 |
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| Mol. Mass. | 359.847 |
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| SMILES | COc1ccc(CCC(=O)N[C@@H](Cc2ccccc2)C(=O)CCl)cc1 |
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| Structure | 
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