| Reaction Details |
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 | Report a problem with these data |
| Target | D(1B) dopamine receptor |
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| Ligand | BDBM50099893 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_61336 |
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| Ki | >10000±n/a nM |
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| Citation |  Huang, Y; Kegeles, LS; Bae, S; Hwang, D; Roth, BL; Savage, JE; Laruelle, M Synthesis of potent and selective dopamine D(4) antagonists as candidate radioligands. Bioorg Med Chem Lett11:1375-7 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1B) dopamine receptor |
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| Name: | D(1B) dopamine receptor |
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| Synonyms: | D(1B) dopamine receptor | DOPAMINE D5 | DRD5_RAT | Dopamine D1B | Dopamine D5 receptor | Dopamine receptor | Drd5 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 52827.88 |
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| Organism: | RAT |
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| Description: | Dopamine D1B 0 RAT::P25115 |
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| Residue: | 475 |
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| Sequence: | MLPPGRNRTAQPARLGLQRQLAQVDAPAGSATPLGPAQVVTAGLLTLLIVWTLLGNVLVC
AAIVRSRHLRAKMTNIFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGTFCDIWVAFDIM
CSTASILNLCIISVDRYWAISRPFRYERKMTQRVALVMVGLAWTLSILISFIPVQLNWHR
DKAGSQGQEGLLSNGTPWEEGWELEGRTENCDSSLNRTYAISSSLISFYIPVAIMIVTYT
RIYRIAQVQIRRISSLERAAEHAQSCRSRGAYEPDPSLRASIKKETKVFKTLSMIMGVFV
CCWLPFFILNCMVPFCSSGDAEGPKTGFPCVSETTFDIFVWFGWANSSLNPIIYAFNADF
RKVFAQLLGCSHFCFRTPVQTVNISNELISYNQDTVFHKEIATAYVHMIPNAVSSGDREV
GEEEEEGPFDHMSQISPTTPDGDLAAESVWELDCEEEVSLGKISPLTPNCFDKTA
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| BDBM50099893 |
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| n/a |
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| Name | BDBM50099893 |
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| Synonyms: | 3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine | CHEMBL28997 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H19FN4 |
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| Mol. Mass. | 310.3687 |
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| SMILES | Fc1ccc(cc1)N1CCN(Cc2c[nH]c3ncccc23)CC1 |
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| Structure | 
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