| Reaction Details |
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 | Report a problem with these data |
| Target | Galectin-8 |
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| Ligand | BDBM50546602 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2016288 (CHEMBL4669866) |
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| Kd | 9170±n/a nM |
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| Citation |  Patel, B; Kishor, C; Houston, TA; Shatz-Azoulay, H; Zick, Y; Vinik, Y; Blanchard, H Rational Design and Synthesis of Methyl-?-d-galactomalonyl Phenyl Esters as Potent Galectin-8 J Med Chem63:11573-11584 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Galectin-8 |
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| Name: | Galectin-8 |
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| Synonyms: | Gal-8 | LEG8_HUMAN | LGALS8 | PCTA-1 | Po66 carbohydrate-binding protein | Po66-CBP | Prostate carcinoma tumor antigen 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 35814.23 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1454625 |
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| Residue: | 317 |
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| Sequence: | MMLSLNNLQNIIYNPVIPFVGTIPDQLDPGTLIVIRGHVPSDADRFQVDLQNGSSMKPRA
DVAFHFNPRFKRAGCIVCNTLINEKWGREEITYDTPFKREKSFEIVIMVLKDKFQVAVNG
KHTLLYGHRIGPEKIDTLGIYGKVNIHSIGFSFSSDLQSTQASSLELTEISRENVPKSGT
PQLRLPFAARLNTPMGPGRTVVVKGEVNANAKSFNVDLLAGKSKDIALHLNPRLNIKAFV
RNSFLQESWGEEERNITSFPFSPGMYFEMIIYCDVREFKVAVNGVHSLEYKHRFKELSSI
DTLEINGDIHLLEVRSW
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| BDBM50546602 |
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| n/a |
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| Name | BDBM50546602 |
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| Synonyms: | CHEMBL4749475 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H22O9 |
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| Mol. Mass. | 370.3512 |
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| SMILES | CO[C@@H]1O[C@H](CO)[C@H](O)[C@H](OC(=O)CC(=O)OCc2ccccc2)[C@H]1O |r| |
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| Structure | 
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