| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50562795 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2080534 (CHEMBL4736325) |
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| Ki | 1330±n/a nM |
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| Citation |  Noguchi, T; Umezaki, Y; Takano, R; Fujimoto, T; Domon, Y; Kubota, K; Ueda, K; Kawase, Y; Yabe, K; Yokoyama, M; Shimada, K A novel [5.2.1]bicyclic amine is a potent analgesic without µ opioid activity. Bioorg Med Chem Lett36:0 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM50562795 |
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| n/a |
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| Name | BDBM50562795 |
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| Synonyms: | CHEMBL4751700 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22N2 |
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| Mol. Mass. | 278.3914 |
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| SMILES | CN1Cc2ccccc2CN2CC[C@]1(C2)c1ccccc1 |r| |
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| Structure | 
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