| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet glycoprotein 4 |
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| Ligand | BDBM50581260 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2150268 (CHEMBL5034730) |
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| IC50 | 670±n/a nM |
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| Citation |  Ohm, RG; Mulumba, M; Chingle, RM; Ahsanullah, na; Zhang, J; Chemtob, S; Ong, H; Lubell, WD Diversity-Oriented A J Med Chem64:9365-9380 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet glycoprotein 4 |
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| Name: | Platelet glycoprotein 4 |
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| Synonyms: | Adipocyte membrane protein | CD36_RAT | CD_antigen=CD36 | Cd36 | Fat | Fatty acid translocase | Fatty acid transport protein | GPIIIB | GPIV | Glycoprotein IIIb | PAS IV | PAS-4 | Platelet glycoprotein IV |
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| Type: | PROTEIN |
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| Mol. Mass.: | 52740.95 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_858884 |
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| Residue: | 472 |
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| Sequence: | MGCDRNCGLITGAVIGAVLAVFGGILMPVGDLLIEKTIKREVVLEEGTIAFKNWVKTGTT
VYRQFWIFDVQNPEEVAKNSSKIKVKQRGPYTYRVRYLAKENITQDPKDSTVSFVQPNGA
IFEPSLSVGTENDNFTVLNLAVAAAPHIYTNSFVQGVLNSLIKKSKSSMFQTRSLKELLW
GYKDPFLSLVPYPISTTVGVFYPYNNTVDGVYKVFNGKDNISKVAIIDTYKGKRNLSYWE
SYCDMINGTDAASFPPFVEKSQTLRFFSSDICRSIYAVFESEVNLKGIPVYRFVLPANAF
ASPLQNPDNHCFCTEKVISNNCTSYGVLDIGKCKEGKPVYISLPHFLHASPDVSEPIEGL
NPNEDEHRTYLDVEPITGFTLQFAKRLQVNILVKPARKIEALKNLKRPYIVPILWLNETG
TIGDEKAEMFRNQVTGKIKLLGLVEMVLLGVGVVMFVAFMISYCACRSKNGK
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| BDBM50581260 |
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| n/a |
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| Name | BDBM50581260 |
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| Synonyms: | CHEMBL4528721 |
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| Type | Small organic molecule |
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| Emp. Form. | C53H64N12O8 |
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| Mol. Mass. | 997.1509 |
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| SMILES | C[C@H](NC(C)=O)C(=O)NN1CC#CCN(CC=C)CCCC[C@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](C)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O)C(N)=O |r| |
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| Structure | 
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