| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
|---|
| Ligand | BDBM50582406 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_2154508 (CHEMBL5039168) |
|---|
| Ki | 0.800000±n/a nM |
|---|
| Citation |  Jiang, S; Iliopoulos-Tsoutsouvas, C; Tong, F; Brust, CA; Keenan, CM; Raghav, JG; Hua, T; Wu, S; Ho, JH; Wu, Y; Grim, TW; Zvonok, N; Thakur, GA; Liu, ZJ; Sharkey, KA; Bohn, LM; Nikas, SP; Makriyannis, A Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists. J Med Chem64:3870-3884 (2021) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 2 |
|---|
| Name: | Cannabinoid receptor 2 |
|---|
| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 38220.43 |
|---|
| Organism: | MOUSE |
|---|
| Description: | P47936 |
|---|
| Residue: | 347 |
|---|
| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
|
|
|
|---|
| BDBM50582406 |
|---|
| n/a |
|---|
| Name | BDBM50582406 |
|---|
| Synonyms: | CHEMBL5091754 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C26H39NO3 |
|---|
| Mol. Mass. | 413.5928 |
|---|
| SMILES | [H][C@@]12C[C@H](CO)CC[C@@]1([H])C(C)(C)Oc1cc(cc(O)c21)C(C)(C)CCCCCCC#N |r| |
|---|
| Structure | 
|
|---|
Search and Browse
