| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50151753 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_305941 |
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| IC50 | 0.180000±n/a nM |
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| Citation |  Weltrowska, G; Lu, Y; Lemieux, C; Chung, NN; Schiller, PW A novel cyclic enkephalin analogue with potent opioid antagonist activity. Bioorg Med Chem Lett14:4731-3 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50151753 |
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| n/a |
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| Name | BDBM50151753 |
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| Synonyms: | 1N-[6-carbamoyl-9-(4-nitrobenzyl)-8,11,14-trioxo-(1R,6S,9S)-3,4-dithia-7,10,13-triazacyclotetradecanyl]-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-(2S)-propanamide | CHEMBL184009 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H35N7O8S2 |
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| Mol. Mass. | 661.75 |
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| SMILES | Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N[C@H]1CSSC[C@@H](NC(=O)[C@H](Cc2ccc(cc2)[N+]([O-])=O)NC(=O)CNC1=O)C(N)=O |
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| Structure | 
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