| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein 5 |
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| Ligand | BDBM50152852 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_305928 (CHEMBL833475) |
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| IC50 | 14000±n/a nM |
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| Citation |  Lehmann, F; Haile, S; Axen, E; Medina, C; Uppenberg, J; Svensson, S; Lundbäck, T; Rondahl, L; Barf, T Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target. Bioorg Med Chem Lett14:4445-8 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein 5 |
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| Name: | Fatty acid-binding protein 5 |
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| Synonyms: | FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 15164.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q01469 |
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| Residue: | 135 |
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| Sequence: | MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
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| BDBM50152852 |
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| n/a |
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| Name | BDBM50152852 |
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| Synonyms: | 3-(5-Bromo-indole-1-sulfonyl)-thiophene-2-carboxylic acid | CHEMBL427320 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H8BrNO4S2 |
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| Mol. Mass. | 386.241 |
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| SMILES | OC(=O)c1sccc1S(=O)(=O)n1ccc2cc(Br)ccc12 |
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| Structure | 
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