| Reaction Details |
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 | Report a problem with these data |
| Target | Protein-lysine 6-oxidase |
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| Ligand | BDBM50589703 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2194162 (CHEMBL5106522) |
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| IC50 | >30000±n/a nM |
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| Citation |  Foot, JS; Buson, A; Deodhar, M; Findlay, AD; Robertson, AD; Turner, CI; Yow, T; Zhou, W; Jarolimek, W Combining monoamine oxidase B and semicarbazide-sensitive amine oxidase enzyme inhibition to address inflammatory disease. Bioorg Med Chem Lett74:0 (2022) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein-lysine 6-oxidase |
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| Name: | Protein-lysine 6-oxidase |
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| Synonyms: | 1.4.3.13 | LOX | LYOX_BOVIN | Lysyl oxidase | Protein-lysine 6-oxidase | Protein-lysine 6-oxidase, long form | Protein-lysine 6-oxidase, short form |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47015.72 |
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| Organism: | Bos taurus |
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| Description: | ChEMBL_118967 |
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| Residue: | 417 |
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| Sequence: | MRFAWTALLGSLQLCALVRCAPPAASHRQPPREQAAAPGAWRQKIQWENNGQVFSLLSLG
SQYQPQRRRDPGATAPGAANATAPQMRTPILLLRNNRTAAARVRTAGPSAAAAGRPRPAA
RHWFQAGYSTSGAHDAGTSRADNQTAPGEVPTLSNLRPPNRVEVDGMVGDDPYNPYKYTD
DNPYYNYYDTYERPRPGSRYRPGYGTGYFQYGLPDLVPDPYYIQASTYVQKMAMYNLRCA
AEENCLASSAYRDVRDYDHRVLLRFPQRVKNQGTSDFLPSRPRYSWEWHSCHQHYHSMDE
FSHYDLLDASTQRRVAEGHKASFCLEDTSCDYGYHRRFACTAHTQGLSPGCYDTYNADID
CQWIDITDVKPGNYILKVSVNPSYLVPESDYSNNVVRCEIRYTGHHAYASGCTISPY
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| BDBM50589703 |
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| n/a |
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| Name | BDBM50589703 |
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| Synonyms: | CHEMBL5196906 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H13ClFNO |
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| Mol. Mass. | 229.678 |
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| SMILES | Cl.NC\C(=C/F)[C@H]1Cc2ccccc2O1 |r| |
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| Structure | 
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