| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50176702 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_327765 (CHEMBL871139) |
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| IC50 | 9.9±n/a nM |
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| Citation |  Mollica, A; Davis, P; Ma, SW; Porreca, F; Lai, J; Hruby, VJ Synthesis and biological activity of the first cyclic biphalin analogues. Bioorg Med Chem Lett16:367-72 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50176702 |
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| n/a |
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| Name | BDBM50176702 |
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| Synonyms: | (S)-2-amino-N-{(4S,10S,15S,21S)-21-[(S)-2-amino-3-(4-hydroxy-phenyl)-propionylamino]-10,15-dibenzyl-5,8,11,14,17,20-hexaoxo-1,2-dithia-6,9,12,13,16,19-hexaaza-cyclodocos-4-yl}-3-(4-hydroxy-phenyl)-propionamide | CHEMBL200129 |
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| Type | Small organic molecule |
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| Emp. Form. | C46H54N10O10S2 |
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| Mol. Mass. | 971.112 |
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| SMILES | N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H]1CSSC[C@@H](NC(=O)[C@@H](N)Cc2ccc(O)cc2)C(=O)NCC(=O)N[C@@H](Cc2ccccc2)C(=O)NNC(=O)[C@H](Cc2ccccc2)NC(=O)CNC1=O |
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| Structure | 
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