| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 1 |
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| Ligand | BDBM50177329 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_329844 (CHEMBL862793) |
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| IC50 | 4660±n/a nM |
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| Citation |  Gududuru, V; Zeng, K; Tsukahara, R; Makarova, N; Fujiwara, Y; Pigg, KR; Baker, DL; Tigyi, G; Miller, DD Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. Bioorg Med Chem Lett16:451-6 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 1 |
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| Name: | Lysophosphatidic acid receptor 1 |
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| Synonyms: | Edg2 | Gpcr91 | LPAR1_RAT | Lpa1 | Lpar1 | Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3 | Lysophosphatidic acid receptor Edg-2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41130.42 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_329844 |
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| Residue: | 364 |
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| Sequence: | MAAASTSSPVISQPQFTAMNEQQCFYNESIAFFYNRSGKYLATEWNTVSKLVMGLGITVC
VFIMLANLLVMVAIYVNRRFHFPIYYLMANLAAADFFAGLAYFYLMFNTGPNTRRLTVST
WLLRQGLIDTSLTASVANLLAIAIERHITVFRMQLHTRMSNRRVVVVIVVIWTMAIVMGA
IPSVGWNCICDIDHCSNMAPLYSDSYLVFWAIFNLVTFVVMVVLYAHIFGYVRQRTMRMS
RHSSGPRRNRDTMMSLLKTVVIVLGAFIVCWTPGLVLLLLDVCCPQCDVLAYEKFFLLLA
EFNSAMNPIIYSYRDKEMSATFRQILCCQRNENPNGPTEGSDRSASSLNHTILAGVHSND
HSVV
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| BDBM50177329 |
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| n/a |
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| Name | BDBM50177329 |
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| Synonyms: | CHEMBL199380 | potassium (2-(6-(4-octylphenyl)hexyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate |
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| Type | Small organic molecule |
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| Emp. Form. | C24H40O6P |
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| Mol. Mass. | 455.5451 |
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| SMILES | CCCCCCCCc1ccc(CCCCCCC2OCC(COP(O)([O-])=O)O2)cc1 |
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| Structure | 
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