| Reaction Details |
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 | Report a problem with these data |
| Target | Proteasome subunit beta type-5 |
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| Ligand | BDBM50185643 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_361596 (CHEMBL868170) |
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| Ki | 18000±n/a nM |
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| Citation |  Basse, N; Papapostolou, D; Pagano, M; Reboud-Ravaux, M; Bernard, E; Felten, AS; Vanderesse, R Development of lipopeptides for inhibiting 20S proteasomes. Bioorg Med Chem Lett16:3277-81 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Proteasome subunit beta type-5 |
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| Name: | Proteasome subunit beta type-5 |
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| Synonyms: | DOA3 | PRE2 | PRG1 | PSB5_YEAST | Proteasome Macropain subunit PRE2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 31634.72 |
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| Organism: | Saccharomyces cerevisiae |
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| Description: | ChEMBL_946840 |
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| Residue: | 287 |
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| Sequence: | MQAIADSFSVPNRLVKELQYDNEQNLESDFVTGASQFQRLAPSLTVPPIASPQQFLRAHT
DDSRNPDCKIKIAHGTTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTM
AGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYT
RKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAA
HRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG
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| BDBM50185643 |
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| n/a |
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| Name | BDBM50185643 |
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| Synonyms: | (S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-(4-hydroxy-phenyl)-propionylamino]-butyrylamino}-4-methyl-pentanoic acid | CHEMBL100097 |
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| Type | Small organic molecule |
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| Emp. Form. | C36H59N3O8 |
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| Mol. Mass. | 661.869 |
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| SMILES | CCCCCCCCCCCCCCCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(O)=O |
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| Structure | 
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