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TargetFatty acid-binding protein, adipocyte
LigandBDBM50192462
Substrate/Competitorn/a
Meas. Tech.ChEMBL_381687 (CHEMBL869163)
Ki 2.5±n/a nM
Citation McDonnell, PAConstantine, KLGoldfarb, VJohnson, SRSulsky, RMagnin, DRRobl, JACaulfield, TJParker, RATaylor, DSAdam, LPMetzler, WJMueller, LFarmer, BT NMR structure of a potent small molecule inhibitor bound to human keratinocyte fatty acid-binding protein. J Med Chem49:5013-7 (2006) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, adipocyte
Name:Fatty acid-binding protein, adipocyte
Synonyms:A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | FABP4 | FABP4_HUMAN | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4 | Fatty acid-binding protein 4 (FABP4)
Type:Enzyme
Mol. Mass.:14719.23
Organism:Homo sapiens (Human)
Description:P15090
Residue:132
Sequence:
MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKN
TEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVM
KGVTSTRVYERA
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  Blast E-value cutoff:
BDBM50192462
n/a
NameBDBM50192462
Synonyms:(S)-2-(2,3-bis(2-chlorobenzyloxy)phenyl)-2-hydroxyacetic acid | CHEMBL378857
TypeSmall organic molecule
Emp. Form.C22H18Cl2O5
Mol. Mass.433.281
SMILESO[C@H](C(O)=O)c1cccc(OCc2ccccc2Cl)c1OCc1ccccc1Cl
Structure
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