| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cholecystokinin receptor type A |
|---|
| Ligand | BDBM50208419 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_443246 (CHEMBL893496) |
|---|
| IC50 | 665±n/a nM |
|---|
| Citation |  Tiwari, AK; Mishra, AK; Bajpai, A; Mishra, P; Singh, S; Sinha, D; Singh, VK Synthesis and evaluation of novel benzimidazole derivative [Bz-Im] and its radio/biological studies. Bioorg Med Chem Lett17:2749-55 (2007) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cholecystokinin receptor type A |
|---|
| Name: | Cholecystokinin receptor type A |
|---|
| Synonyms: | CCKAR_RAT | Cckar | Cholecystokinin peripheral | Cholecystokinin receptor | Cholecystokinin receptor type A |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 49676.37 |
|---|
| Organism: | RAT |
|---|
| Description: | Cholecystokinin central 0 RAT::P30551 |
|---|
| Residue: | 444 |
|---|
| Sequence: | MSHSPARQHLVESSRMDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSALQI
LLYSIIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLK
DFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAAT
WCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLLPGIVM
VVAYGLISLELYQGIKFDASQKKSAKEKKPSTGSSTRYEDSDGCYLQKSRPPRKLELQQL
SSGSGGSRLNRIRSSSSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAE
KHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPPGVRGEVGEEE
DGRTIRALLSRYSYSHMSTSAPPP
|
|
|
|---|
| BDBM50208419 |
|---|
| n/a |
|---|
| Name | BDBM50208419 |
|---|
| Synonyms: | 2-{2-hydroxy-5-[(E)-2-(4-hydroxy-phenyl)-vinyl]-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl}-isoindole-1,3-dione | CHEMBL389311 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C32H21N3O4 |
|---|
| Mol. Mass. | 511.5268 |
|---|
| SMILES | Oc1ccc(\C=C\c2cc3nc4ccccc4n3c3c(CN4C(=O)c5ccccc5C4=O)c(O)ccc23)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
