| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
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| Ligand | BDBM50227099 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_452341 (CHEMBL902578) |
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| Ki | >10000±n/a nM |
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| Citation |  Martin, RE; Green, LG; Guba, W; Kratochwil, N; Christ, A Discovery of the first nonpeptidic, small-molecule, highly selective somatostatin receptor subtype 5 antagonists: a chemogenomics approach. J Med Chem50:6291-4 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 1 |
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| Name: | Somatostatin receptor type 1 |
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| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42692.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30872 |
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| Residue: | 391 |
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| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
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| BDBM50227099 |
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| n/a |
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| Name | BDBM50227099 |
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| Synonyms: | 2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide | CHEMBL236788 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H31N5O5S |
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| Mol. Mass. | 489.588 |
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| SMILES | CCOc1cc(CN2CCC(CC2)Nc2nc3cc(ccc3o2)S(N)(=O)=O)cc(OCC)c1N |
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| Structure | 
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