| Reaction Details |
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 | Report a problem with these data |
| Target | Type-1 angiotensin II receptor |
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| Ligand | BDBM50251488 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_488661 (CHEMBL988351) |
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| Ki | 3±n/a nM |
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| Citation |  Wallinder, C; Botros, M; Rosenström, U; Guimond, MO; Beaudry, H; Nyberg, F; Gallo-Payet, N; Hallberg, A; Alterman, M Selective angiotensin II AT2 receptor agonists: Benzamide structure-activity relationships. Bioorg Med Chem16:6841-9 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Type-1 angiotensin II receptor |
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| Name: | Type-1 angiotensin II receptor |
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| Synonyms: | AGTR1 | AGTR1_PIG |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40925.99 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_488661 |
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| Residue: | 359 |
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| Sequence: | MILNSSTEDSIKRIQDDCPKAGRHNYIFVMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLK
TVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNYLCKIASASVSFNLYASVFLLT
CLSIDRYLAIVHPMKSRLRRTMLVAKVTCIIIWLLAGLASLPTIIHRNVFFIENTNITVC
AFHYESQNSTLPVGLGLTKNILGFLFPFLIILTSYTLIWKALKKAYEIQKNKPRNDDIFK
IIMAIVLFFFFSWVPHQIFTFLDVLIQLGIIHDCKIADIVDTAMPITICLAYFNNCLNPL
FYGFLGKKFKKYFLQLLKYIPPKAKSHSSLSTKMSTLSYRPSENGSSSTKKSAPCTEVE
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| BDBM50251488 |
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| n/a |
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| Name | BDBM50251488 |
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| Synonyms: | CHEMBL521093 | N-Butoxycarbonyl-3-[4-(N,N-diethylcarbamoyl)phenyl]-5-isobutylthiophene-2-sulfonamide |
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| Type | Small organic molecule |
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| Emp. Form. | C24H34N2O5S2 |
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| Mol. Mass. | 494.667 |
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| SMILES | CCCCOC(=O)NS(=O)(=O)c1sc(CC(C)C)cc1-c1ccc(cc1)C(=O)N(CC)CC |
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| Structure | 
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