| Reaction Details |
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 | Report a problem with these data |
| Target | Type-1 angiotensin II receptor |
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| Ligand | BDBM50141059 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_488661 (CHEMBL988351) |
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| Ki | 0.7±n/a nM |
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| Citation |  Wallinder, C; Botros, M; Rosenström, U; Guimond, MO; Beaudry, H; Nyberg, F; Gallo-Payet, N; Hallberg, A; Alterman, M Selective angiotensin II AT2 receptor agonists: Benzamide structure-activity relationships. Bioorg Med Chem16:6841-9 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Type-1 angiotensin II receptor |
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| Name: | Type-1 angiotensin II receptor |
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| Synonyms: | AGTR1 | AGTR1_PIG |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40925.99 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_488661 |
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| Residue: | 359 |
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| Sequence: | MILNSSTEDSIKRIQDDCPKAGRHNYIFVMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLK
TVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNYLCKIASASVSFNLYASVFLLT
CLSIDRYLAIVHPMKSRLRRTMLVAKVTCIIIWLLAGLASLPTIIHRNVFFIENTNITVC
AFHYESQNSTLPVGLGLTKNILGFLFPFLIILTSYTLIWKALKKAYEIQKNKPRNDDIFK
IIMAIVLFFFFSWVPHQIFTFLDVLIQLGIIHDCKIADIVDTAMPITICLAYFNNCLNPL
FYGFLGKKFKKYFLQLLKYIPPKAKSHSSLSTKMSTLSYRPSENGSSSTKKSAPCTEVE
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| BDBM50141059 |
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| n/a |
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| Name | BDBM50141059 |
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| Synonyms: | CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-5-isobutyl-biphenyl-2-sulfonic acid amide |
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| Type | Small organic molecule |
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| Emp. Form. | C32H40N4O4S |
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| Mol. Mass. | 576.749 |
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| SMILES | CCCCOC(=O)NS(=O)(=O)c1ccc(CC(C)C)cc1-c1ccc(Cn2c(CC)nc3c(C)cc(C)nc23)cc1 |
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| Structure | 
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