| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Disks large homolog 4 |
|---|
| Ligand | BDBM50252746 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_539187 (CHEMBL1024691) |
|---|
| Ki | 69000±n/a nM |
|---|
| Citation |  Bach, A; Chi, CN; Olsen, TB; Pedersen, SW; Røder, MU; Pang, GF; Clausen, RP; Jemth, P; Strømgaard, K Modified peptides as potent inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction. J Med Chem51:6450-9 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Disks large homolog 4 |
|---|
| Name: | Disks large homolog 4 |
|---|
| Synonyms: | DLG4 | DLG4_HUMAN | PSD95 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 80483.80 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_736705 |
|---|
| Residue: | 724 |
|---|
| Sequence: | MDCLCIVTTKKYRYQDEDTPPLEHSPAHLPNQANSPPVIVNTDTLEAPGYELQVNGTEGE
MEYEEITLERGNSGLGFSIAGGTDNPHIGDDPSIFITKIIPGGAAAQDGRLRVNDSILFV
NEVDVREVTHSAAVEALKEAGSIVRLYVMRRKPPAEKVMEIKLIKGPKGLGFSIAGGVGN
QHIPGDNSIYVTKIIEGGAAHKDGRLQIGDKILAVNSVGLEDVMHEDAVAALKNTYDVVY
LKVAKPSNAYLSDSYAPPDITTSYSQHLDNEISHSSYLGTDYPTAMTPTSPRRYSPVAKD
LLGEEDIPREPRRIVIHRGSTGLGFNIVGGEDGEGIFISFILAGGPADLSGELRKGDQIL
SVNGVDLRNASHEQAAIALKNAGQTVTIIAQYKPEEYSRFEAKIHDLREQLMNSSLGSGT
ASLRSNPKRGFYIRALFDYDKTKDCGFLSQALSFRFGDVLHVIDASDEEWWQARRVHSDS
ETDDIGFIPSKRRVERREWSRLKAKDWGSSSGSQGREDSVLSYETVTQMEVHYARPIIIL
GPTKDRANDDLLSEFPDKFGSCVPHTTRPKREYEIDGRDYHFVSSREKMEKDIQAHKFIE
AGQYNSHLYGTSVQSVREVAEQGKHCILDVSANAVRRLQAAHLHPIAIFIRPRSLENVLE
INKRITEEQARKAFDRATKLEQEFTECFSAIVEGDSFEEIYHKVKRVIEDLSGPYIWVPA
RERL
|
|
|
|---|
| BDBM50252746 |
|---|
| n/a |
|---|
| Name | BDBM50252746 |
|---|
| Synonyms: | CHEMBL492431 | N-Ethyl-ETAV |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H34N4O8 |
|---|
| Mol. Mass. | 446.4953 |
|---|
| SMILES | CCN[C@@H](CCC(O)=O)C(=O)N[C@@H](C(C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(O)=O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
