Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194124 ((S)-N-(1-(5-(6-aminohexylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122077 (CHEMBL153017 | N-[1-[5-(6-Amino-hexylamino)-pentyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194124 ((S)-N-(1-(5-(6-aminohexylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194127 ((S)-N-(1-(5-(7-aminoheptylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194123 ((S)-N-(1-(5-(5-aminopentylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194113 ((S)-N-(1-(5-(4-aminobutylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194118 ((S)-N-(1-(5-(3-aminopropylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194111 ((S)-N-(1-(5-(10-aminodecylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194109 ((S)-N-(1-(5-(8-aminooctylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194114 ((S)-N-(1-(9-(6-aminohexylamino)nonylamino)-3-(4-hy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194119 ((S)-N-(1-(4-(7-aminoheptylamino)butylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122093 (CHEMBL152879 | N-[1-[4-(7-Amino-heptylamino)-butyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194120 ((S)-N-(1-(4-(6-aminohexylamino)butylamino)-3-(4-hy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194118 ((S)-N-(1-(5-(3-aminopropylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122084 (CHEMBL153996 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194117 ((S)-N-(1-(5-(9-aminononylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194122 ((S)-N-(1-(8-(3-aminopropylamino)octylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122090 (CHEMBL147182 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194113 ((S)-N-(1-(5-(4-aminobutylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 68 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122096 (CHEMBL152410 | Hexanoic acid [1-[8-(3-amino-propyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 68 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194126 ((S)-N-(1-(8-(6-aminohexylamino)octylamino)-3-(4-hy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 77 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194112 ((S)-N-(1-(5-(12-aminododecylamino)pentylamino)-3-(...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 77 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122087 (CHEMBL153995 | Cyclohexanecarboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122085 (CHEMBL152425 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118202 (6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122086 (CHEMBL269192 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194123 ((S)-N-(1-(5-(5-aminopentylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123637 (6-benzyloxy-8-(tert-butyl)-9-flouro-12,17-dihydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122095 (CHEMBL355977 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123639 (8-(tert-butyl)-9-chloro-6,12,17-trihydroxy-16-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122092 (CHEMBL350228 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122091 (CHEMBL152736 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194127 ((S)-N-(1-(5-(7-aminoheptylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123644 (6-benzyloxy-8-(tert-butyl)-12,17-dihydroxy-16-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194116 ((S)-N-(1-(3-(6-aminohexylamino)propylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118204 (6-(4-benzoylphenylcarbonyloxy)-8-(tert-butyl)-12,1...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122094 (CHEMBL345521 | Pyridine-2-carboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122089 (CHEMBL352030 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122093 (CHEMBL152879 | N-[1-[4-(7-Amino-heptylamino)-butyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194115 ((S)-N-(1-(5-(2-aminoethylamino)pentylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122086 (CHEMBL269192 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118194 (8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-t...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118201 (6-(4-benzoylbenzyloxy)-8-(tert-butyl)-12,17-dihydr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194110 ((S)-N-(1-(7-(4-aminobutylamino)heptylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 168 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122078 (CHEMBL422515 | N-[1-[7-(4-Amino-butylamino)-heptyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 168 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122094 (CHEMBL345521 | Pyridine-2-carboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122091 (CHEMBL152736 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194111 ((S)-N-(1-(5-(10-aminodecylamino)pentylamino)-3-(4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194108 ((S)-N-(1-(2-(6-aminohexylamino)ethylamino)-3-(4-hy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 208 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Rattus norvegicus (Rat)) | BDBM50194107 ((S)-N-(1-(7-(6-aminohexylamino)heptylamino)-3-(4-h...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 208 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences Curated by ChEMBL | Assay Description Antagonist activity against rat GluR1 flop expressed in Xenopus laevis oocyte assessed as inhibition of glutamate-induced current at holding potentia... | J Med Chem 49: 5414-23 (2006) Article DOI: 10.1021/jm060606j BindingDB Entry DOI: 10.7270/Q24X57FS | |||||||||||
More data for this Ligand-Target Pair |
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