| Reaction Details |
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 | Report a problem with these data |
| Target | Peroxisome proliferator-activated receptor delta |
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| Ligand | BDBM50246088 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_558114 (CHEMBL959043) |
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| EC50 | >25000±n/a nM |
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| Citation |  Martres, P; Faucher, N; Laroze, A; Pineau, O; Fouchet, MH; Potvain, F; Grillot, D; Beneton, V The discovery of equipotent PPARalpha/gamma dual activators. Bioorg Med Chem Lett18:6251-4 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Peroxisome proliferator-activated receptor delta |
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| Name: | Peroxisome proliferator-activated receptor delta |
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| Synonyms: | NUC1 | Nr1c2 | Nuclear hormone receptor 1 | Nuclear receptor subfamily 1 group C member 2 | PPAR-beta | PPAR-delta | PPARD_MOUSE | Pparb | Ppard |
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| Type: | PROTEIN |
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| Mol. Mass.: | 49719.14 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_1288931 |
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| Residue: | 440 |
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| Sequence: | MEQPQEETPEAREEEKEEVAMGDGAPELNGGPEHTLPSSSCADLSQNSSPSSLLDQLQMG
CDGASGGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCDRICKIQKKN
RNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTASEGCQHNPQLADLKAFSKH
IYNAYLKNFNMTKKKARSILTGKSSHNAPFVIHDIETLWQAEKGLVWKQLVNGLPPYNEI
SVHVFYRCQSTTVETVRELTEFAKNIPNFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKD
GLLVANGSGFVTHEFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDR
PGLMNVPQVEAIQDTILRALEFHLQVNHPDSQYLFPKLLQKMADLRQLVTEHAQMMQWLK
KTESETLLHPLLQEIYKDMY
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| BDBM50246088 |
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| n/a |
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| Name | BDBM50246088 |
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| Synonyms: | 2-methyl-2-[2-methyl-4-({[1-methyl-5-(2'-methyl-biphenyl-4-yl)-1H-pyrazole-3-carbonyl]-amino}-methyl)-phenoxy]-propionic acid | CHEMBL472399 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H31N3O4 |
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| Mol. Mass. | 497.5848 |
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| SMILES | Cc1cc(CNC(=O)c2cc(-c3ccc(cc3)-c3ccccc3C)n(C)n2)ccc1OC(C)(C)C(O)=O |
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| Structure | 
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