| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein kinase 17A |
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| Ligand | BDBM50273636 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_537119 (CHEMBL988951) |
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| Kd | 96±n/a nM |
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| Citation |  Bamborough, P; Drewry, D; Harper, G; Smith, GK; Schneider, K Assessment of chemical coverage of kinome space and its implications for kinase drug discovery. J Med Chem51:7898-914 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Serine/threonine-protein kinase 17A |
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| Name: | Serine/threonine-protein kinase 17A |
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| Synonyms: | DRAK1 | ST17A_HUMAN | STK17A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 46544.04 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_109255245 |
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| Residue: | 414 |
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| Sequence: | MIPLEKPGSGGSSPGATSGSGRAGRGLSGPCRPPPPPQARGLLTEIRAVVRTEPFQDGYS
LCPGRELGRGKFAVVRKCIKKDSGKEFAAKFMRKRRKGQDCRMEIIHEIAVLELAQDNPW
VINLHEVYETASEMILVLEYAAGGEIFDQCVADREEAFKEKDVQRLMRQILEGVHFLHTR
DVVHLDLKPQNILLTSESPLGDIKIVDFGLSRILKNSEELREIMGTPEYVAPEILSYDPI
SMATDMWSIGVLTYVMLTGISPFLGNDKQETFLNISQMNLSYSEEEFDVLSESAVDFIRT
LLVKKPEDRATAEECLKHPWLTQSSIQEPSFRMEKALEEANALQEGHSVPEINSDTDKSE
TKESIVTEELIVVTSYTLGQCRQSEKEKMEQKAISKRFKFEEPLLQEIPGEFIY
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| BDBM50273636 |
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| n/a |
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| Name | BDBM50273636 |
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| Synonyms: | 4-(5-(4-fluorophenyl)-1H-pyrazol-3-ylamino)benzamide | CHEMBL511337 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13FN4O |
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| Mol. Mass. | 296.299 |
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| SMILES | NC(=O)c1ccc(Nc2cc(n[nH]2)-c2ccc(F)cc2)cc1 |
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| Structure | 
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