| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Serine/threonine-protein kinase Nek7 |
|---|
| Ligand | BDBM50273636 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_537120 (CHEMBL988952) |
|---|
| Kd | >40000±n/a nM |
|---|
| Citation |  Bamborough, P; Drewry, D; Harper, G; Smith, GK; Schneider, K Assessment of chemical coverage of kinome space and its implications for kinase drug discovery. J Med Chem51:7898-914 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Serine/threonine-protein kinase Nek7 |
|---|
| Name: | Serine/threonine-protein kinase Nek7 |
|---|
| Synonyms: | NEK kinase | NEK7 | NEK7_HUMAN |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 34559.15 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_586832 |
|---|
| Residue: | 302 |
|---|
| Sequence: | MDEQSQGMQGPPVPQFQPQKALRPDMGYNTLANFRIEKKIGRGQFSEVYRAACLLDGVPV
ALKKVQIFDLMDAKARADCIKEIDLLKQLNHPNVIKYYASFIEDNELNIVLELADAGDLS
RMIKHFKKQKRLIPERTVWKYFVQLCSALEHMHSRRVMHRDIKPANVFITATGVVKLGDL
GLGRFFSSKTTAAHSLVGTPYYMSPERIHENGYNFKSDIWSLGCLLYEMAALQSPFYGDK
MNLYSLCKKIEQCDYPPLPSDHYSEELRQLVNMCINPDPEKRPDVTYVYDVAKRMHACTA
SS
|
|
|
|---|
| BDBM50273636 |
|---|
| n/a |
|---|
| Name | BDBM50273636 |
|---|
| Synonyms: | 4-(5-(4-fluorophenyl)-1H-pyrazol-3-ylamino)benzamide | CHEMBL511337 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H13FN4O |
|---|
| Mol. Mass. | 296.299 |
|---|
| SMILES | NC(=O)c1ccc(Nc2cc(n[nH]2)-c2ccc(F)cc2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
