Reaction Details |
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Target | Serine/threonine-protein kinase 16 |
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Ligand | BDBM50273541 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_537068 (CHEMBL986217) |
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Kd | 24±n/a nM |
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Citation | Bamborough, P; Drewry, D; Harper, G; Smith, GK; Schneider, K Assessment of chemical coverage of kinome space and its implications for kinase drug discovery. J Med Chem51:7898-914 (2008) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Serine/threonine-protein kinase 16 |
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Name: | Serine/threonine-protein kinase 16 |
Synonyms: | MPSK1 | PKL12 | STK16 | STK16_HUMAN | Serine/threonine-protein kinase 16 | TSF1 | Tyrosine-protein kinase STK16 (STK16) |
Type: | Protein |
Mol. Mass.: | 34659.07 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 305 |
Sequence: | MGHALCVCSRGTVIIDNKRYLFIQKLGEGGFSYVDLVEGLHDGHFYALKRILCHEQQDRE
EAQREADMHRLFNHPNILRLVAYCLRERGAKHEAWLLLPFFKRGTLWNEIERLKDKGNFL
TEDQILWLLLGICRGLEAIHAKGYAHRDLKPTNILLGDEGQPVLMDLGSMNQACIHVEGS
RQALTLQDWAAQRCTISYRAPELFSVQSHCVIDERTDVWSLGCVLYAMMFGEGPYDMVFQ
KGDSVALAVQNQLSIPQSPRHSSALRQLLNSMMTVDPHQRPHIPLLLSQLEALQPPAPGQ
HTTQI
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BDBM50273541 |
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n/a |
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Name | BDBM50273541 |
Synonyms: | CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)nicotinamide |
Type | Small organic molecule |
Emp. Form. | C20H13N5O |
Mol. Mass. | 339.3501 |
SMILES | O=C(Nc1c[nH]c2ncc(cc12)-c1ccc(cc1)C#N)c1cccnc1 |
Structure |
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