| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Retinoic acid receptor gamma |
|---|
| Ligand | BDBM50265918 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_540171 (CHEMBL1029012) |
|---|
| EC50 | >1000±n/a nM |
|---|
| Citation |  Charton, J; Deprez-Poulain, R; Hennuyer, N; Tailleux, A; Staels, B; Deprez, B Novel non-carboxylic acid retinoids: 1,2,4-oxadiazol-5-one derivatives. Bioorg Med Chem Lett19:489-92 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Retinoic acid receptor gamma |
|---|
| Name: | Retinoic acid receptor gamma |
|---|
| Synonyms: | NR1B3 | Nuclear receptor subfamily 1 group B member 3 | RAR-gamma | RARG | RARG_HUMAN | Retinoic acid receptor RXR-alpha/gamma | Retinoic acid receptor gamma | Retinoid receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 50345.43 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1458016 |
|---|
| Residue: | 454 |
|---|
| Sequence: | MATNKERLFAAGALGPGSGYPGAGFPFAFPGALRGSPPFEMLSPSFRGLGQPDLPKEMAS
LSVETQSTSSEEMVPSSPSPPPPPRVYKPCFVCNDKSSGYHYGVSSCEGCKGFFRRSIQK
NMVYTCHRDKNCIINKVTRNRCQYCRLQKCFEVGMSKEAVRNDRNKKKKEVKEEGSPDSY
ELSPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIK
IVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMH
NAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEA
LRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLENPE
MFEDDSSQPGPHPNASSEDEVPGGQGKGGLKSPA
|
|
|
|---|
| BDBM50265918 |
|---|
| n/a |
|---|
| Name | BDBM50265918 |
|---|
| Synonyms: | 3-(4-((4-tert-butylphenyl)ethynyl)phenyl)-1,2,4-oxadiazol-5(4H)-one | CHEMBL511855 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H18N2O2 |
|---|
| Mol. Mass. | 318.3691 |
|---|
| SMILES | CC(C)(C)c1ccc(cc1)C#Cc1ccc(cc1)-c1nc(=O)o[nH]1 |
|---|
| Structure | 
|
|---|
Search and Browse
