| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 4 |
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| Ligand | BDBM29526 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_3341 (CHEMBL619041) |
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| Ki | 1.07±n/a nM |
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| Citation |  Langlois, M; Zhang, L; Bre´mont, B; Shen, S; Manara, L; Croci, T Design of a potent 5-HT4 receptor agonist with nanomolar affinity Bioorg Med Chem Lett4:1433-1436 (1994) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 4 |
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| Name: | 5-hydroxytryptamine receptor 4 |
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| Synonyms: | 5-HT-4 | 5-HT4 | 5-HT4L | 5-HT4S | 5-hydroxytryptamine receptor 4 | 5HT4R_RAT | Htr4 | Serotonin (5-HT) receptor | Serotonin 4 (5-HT4) receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 46117.31 |
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| Organism: | RAT |
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| Description: | 5-HT4 HTR4 RAT::Q62758 |
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| Residue: | 406 |
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| Sequence: | MDRLDANVSSNEGFGSVEKVVLLTFFAMVILMAILGNLLVMVAVCRDRQLRKIKTNYFIV
SLAFADLLVSVLVNAFGAIELVQDIWFYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYY
AICCQPLVYRNKMTPLRIALMLGGCWVIPMFISFLPIMQGWNNIGIVDVIEKRKFNHNSN
STFCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRP
QTADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEKVWTAFLWL
GYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRD
TVECGGQWESRCHLTATSPLVAAQPVIRRPQDNDLEDSCSLKRSQS
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| BDBM29526 |
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| n/a |
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| Name | BDBM29526 |
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| Synonyms: | 2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoate | CHEMBL286136 | ML 10302 | ML10302 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H21ClN2O3 |
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| Mol. Mass. | 312.792 |
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| SMILES | COc1cc(N)c(Cl)cc1C(=O)OCCN1CCCCC1 |
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| Structure | 
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