| Reaction Details |
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 | Report a problem with these data |
| Target | Gastrin/cholecystokinin type B receptor |
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| Ligand | BDBM50283961 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_49416 (CHEMBL658776) |
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| IC50 | 8500±n/a nM |
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| Citation |  Horwell, DC; Lennon, IC; Roberts, E Alternative strategies towards the identification of chemical lead compounds by rational design Bioorg Med Chem Lett4:525-530 (1994) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Gastrin/cholecystokinin type B receptor |
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| Name: | Gastrin/cholecystokinin type B receptor |
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| Synonyms: | Cckbr | Cholecystokinin A | Cholecystokinin receptor | GASR_MOUSE | Gastrin/cholecystokinin type B receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 49196.59 |
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| Organism: | MOUSE |
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| Description: | Cholecystokinin A CCKBR MOUSE::P56481 |
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| Residue: | 453 |
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| Sequence: | MDLLKLNRSLQGPGPGSGSSLCRPGVSLLNSSSAGNLSCETPRIRGTGTRELELTIRITL
YAVIFLMSVGGNVLIIVVLGLSRRLRTVTNAFLLSLAVSDLLLAVACMPFTLLPNLMGTF
IFGTVICKAVSYLMGVSVSVSTLNLAAIALERYSAICRPLQARVWQTRSHAARVILATWL
LSGLLMVPYPVYTVVQPVGPRILQCMHLWPSERVQQMWSVLLLILLFFIPGVVMAVAYGL
ISRELYLGLRFDGDNDSETQSRVRNQGGLPGGAAAPGPVHQNGGCRHVTSLTGEDSDGCY
VQLPRSRLEMTTLTTPTTGPGPGPRPNQAKLLAKKRVVRMLLVIVLLFFVCWLPVYSANT
WRAFDGPGARRALAGAPISFIHLLSYTSACANPLVYCFMHRRFRQACLDTCARCCPRPPR
ARPRPLPDEDPPTPSIASLSRLSYTTISTLGPG
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| BDBM50283961 |
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| n/a |
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| Name | BDBM50283961 |
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| Synonyms: | 3-[1-Benzyl-4-(diethoxy-phosphoryloxy)-1,2,3,6-tetrahydro-pyridin-3-ylmethyl]-indole-1-carboxylic acid tert-butyl ester | CHEMBL151022 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H39N2O6P |
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| Mol. Mass. | 554.6142 |
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| SMILES | CCOP(=O)(OCC)OC1=CCN(Cc2ccccc2)CC1Cc1cn(C(=O)OC(C)(C)C)c2ccccc12 |t:9| |
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| Structure | 
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