| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50287931 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_46461 |
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| Ki | >20000±n/a nM |
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| Citation |  Gareau, Y; Dufresne, C; Gallant, M; Rochette, C; Sawyer, N; Slipetz, DM; Tremblay, N; Weech, PK; Metters, KM; Labelle, M Structure activity relationships of tetrahydrocannabinol analogues on human cannabinoid receptors Bioorg Med Chem Lett6:189-194 (1996) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52868.96 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21554 |
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| Residue: | 472 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50287931 |
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| n/a |
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| Name | BDBM50287931 |
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| Synonyms: | 4-(1,1-Dimethyl-heptyl)-2,6-dimethoxy-3',5'-dimethyl-biphenyl | CHEMBL61037 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H36O2 |
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| Mol. Mass. | 368.5521 |
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| SMILES | CCCCCCC(C)(C)c1cc(OC)c(c(OC)c1)-c1cc(C)cc(C)c1 |
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| Structure | 
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